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AxisPharm provides high purity PROTAC PEG reagents (linkers) with various active groups, such as azide, acid, amine, etc.
The design of Proteolysis Targeting Chimera (PROTACs) is a powerful small molecule approach for inducing protein degradation for anticancer therapy. PROTACs conjugate a target warhead to an E3 ubiquitin ligase ligand via a linker. To further empower the PROTAC study, AxisPharm are developing a series of PROTAC linker to accelerate our customers’  R&D effort.

Cat# Name Structure M.W. Purity Pricing
(S,R,S)-AHPC-amido-acid
AP14172(S,R,S)-AHPC-amido-C2-acid530.60≥95% Pricing
AP14171(S,R,S)-AHPC-amido-C6-acid586.80≥95% Pricing
(S,R,S)-AHPC-Boc
AP14173(S,R,S)-AHPC-Boc530.70≥95% Pricing
(S,R,S)-AHPC-Me-amine
AP14168(S,R,S)-AHPC-Me-C10-NH2627.90≥95% Pricing
(S,R. S)-AHPC-PEG-acid
AP13442(S,R,S)-AHPC-pentanoic-acid558.7≥98% Pricing
AP14164(S, R, S)-AHPC-nanoly-acid614.80≥95% Pricing
AP12132(S,R. S)-AHPC-PEG2-acid618.75≥95% Pricing
AP13438(S,R,S)-AHPC-PEG3-acid662.8≥98% Pricing
AP13439(S,R,S)-AHPC-PEG4-acid706.9≥98% Pricing
AP13440(S,R,S)-AHPC-PEG6-acid795≥98% Pricing
AP13441(S,R,S)-AHPC-PEG8-acid883≥98% Pricing
(S,R. S)-AHPC-PEG-amine
AP14170(S,R,S)-AHPC-C4-NH2529.70≥95% Pricing
AP14169(S,R,S)-AHPC-C6-NH2557.80≥95% Pricing
AP12133(S,R. S)-AHPC-PEG2-amine hydrochloride salt575.73≥95% Pricing
AP13954(S, R, S)-AHPC-PEG3-amine hydrochloride salt619.8≥95% Pricing
AP12134(S,R. S)-AHPC-PEG4-amine hydrochloride salt663.83≥95% Pricing
(S,R. S)-AHPC-PEG-Azide
AP12135(S,R. S)-AHPC-PEG4-Azide703.86≥95% Pricing
(S,R. S)-AHPC-PEG-NHS ester
AP13391(S,R,S)-AHPC-PEG2-NHS ester715.8≥98% Pricing
AP13392(S,R,S)-AHPC-PEG4-NHS ester803.9≥98% Pricing
AP13403(S,R,S)-AHPC-PEG6-NHS ester892≥95% Pricing
AP13404(S,R,S)-AHPC-PEG8-NHS ester980.2≥98% Pricing
(S,R. S)-AHPC-PEG-tosyl
AP14165(S, R, S)-AHPC-PEG2-Tos700.90≥95% Pricing
AP14166(S, R, S)-AHPC-PEG4-tosyl789.00≥95% Pricing
AP14167(S, R, S)-AHPC-PEG6-Tos877.10≥95% Pricing
4-Fluoro-thalidomide
AP121294-Fluoro-thalidomide276.22≥95% Pricing
4-Hydroxy-thalidomide
AP121224-Hydroxy-thalidomide274.23≥95% Pricing
ARV-110
AP14691ARV-110812.30≥95% Pricing
ARV-825
AP14692ARV-825923.5≥95% Pricing
BET Inhibitors
AP14266PFI 3321.40≥95% Pricing
AP14265PFI 1347.40≥95% Pricing
AP14256BI 9564353.40≥95% Pricing
AP14255BAZ2-ICR357.40≥95% Pricing
AP14253RVX-208370.40≥95% Pricing
AP14259GSK 2801371.50≥95% Pricing
AP14267PFI 4380.50≥95% Pricing
AP14251MS-436383.40≥95% Pricing
AP14263NI 57383.40≥95% Pricing
AP14260GSK 5959394.50≥95% Pricing
AP14258CPI 203399.90≥95% Pricing
AP14257Bromosporine404.50≥95% Pricing
AP14261GSK 6853409.50≥95% Pricing
AP14250I-BET 762423.90≥95% Pricing
AP14254BAY 299429.50≥95% Pricing
AP14272l-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)-lHpyrazolo [3,4-d]pyrimidin-l-yl]-l-piperidinyl]-2-propyn-l-one438.50≥95% Pricing
AP14249(+)JQ-1457.00≥95% Pricing
AP142734-(4-(4-(3-fluorobenzyloxy)-3-chlorophenylamino)quinazolin-6-yl)phenol471.90≥95% Pricing
AP14269XMD 8-92474.60≥95% Pricing
AP14264OTX 015492.00≥95% Pricing
AP14262I-BRD9497.60≥95% Pricing
AP14270N-[3-Chloro-4-(3-fluorobenzyloxy)phenyl]-6-iodoquinazolin-4-amine505.70≥95% Pricing
AP14268SGC-CBP30509.10≥95% Pricing
AP14252BI-2536521.70≥95% Pricing
AP14271dBET1785.3≥95% Pricing
BETd-260
AP14690BETd-260798.90≥95% Pricing
BTK kinase inhibitor
AP14294IBT6A386.50≥95% Pricing
CFT7455
AP15056CFT7455469.5≥95% Pricing
E3 Ligand
AP14275LCL161500.60≥95% Pricing
AP14277Nutlin-3581.50≥95% Pricing
AP14276Idasanutlin616.50≥95% Pricing
E3 Ligase ligand
AP14439E3 Ligase ligand 9408.50≥95% Pricing
AP14437E3 Ligase ligand 1a444.60≥95% Pricing
AP14438E3 ligase Ligand 19532.60≥95% Pricing
Iberdomide
AP15055Iberdomide449.5≥95% Pricing
Lenalidomide
AP13829Phthalimidine, 2-(2,6-dioxopiperiden-3-yl)244.3≥95% Pricing
AP139693-(7-Amino-1-oxoisoindolin-2-yl)piperidine-2,6-dione259.26≥95% Pricing
AP139703-(6-Amino-1-oxoisoindolin-2-yl)piperidine-2,6-dione259.26≥95% Pricing
AP139683-(5-Amino-1-oxoisoindolin-2-yl)piperidine-2,6-dione259.26≥95% Pricing
AP13967Lenalidomide259.26≥95% Pricing
AP13977Lenalidomide-OH260.30≥95% Pricing
AP137302-(2,6-Dioxopiperidin-3-yl)-1-oxoisoindoline-5-carboxylic acid288.3≥95% Pricing
AP137312-(2,6-dioxopiperidin-3-yl)-1-oxo-2,3-dihydro-1H-isoindole-4-carboxylic acid288.3≥95% Pricing
AP139713-(5-(Aminomethyl)-1-oxoisoindolin-2-yl)piperidine-2,6-dione hydrochloride309.75≥95% Pricing
AP139733-(5-Bromo-1-oxo-2-isoindolinyl)piperidine-2,6-dione323.14≥95% Pricing
AP139753-(6-Bromo-1-oxoisoindolin-2-yl)piperidine-2,6-dione323.14≥95% Pricing
AP139723-(4-Bromo-1-oxoisoindolin-2-yl)piperidine-2,6-dione323.14≥95% Pricing
AP139743-(7-Bromo-1-oxoisoindolin-2-yl)piperidine-2,6-dione323.14≥95% Pricing
AP139763-(5-iodo-1-oxo-2,3-dihydro-1H-isoindol-2-yl)piperidine-2,6-dione370.14≥95% Pricing
MZ1
AP14307ARV-771986.70≥95% Pricing
AP14308MZ11002.6≥95% Pricing
Pomalidomide
AP13277Pomalidomide273.2≥98% Pricing
Pomalidomide-PEG-Acid
AP12995Pomalidomide-PEG3-Acid477.47≥95% Pricing
AP12396Pomalidomide-PEG4-Acid521.52≥95% Pricing
AP13000Pomalidomide-PEG5-Acid565.58≥95% Pricing
Pomalidomide-PEG-Amine
AP13888Pomalidomide-PEG3-Amine HCl salt484.9≥95% Pricing
Pomalidomide-PEG-Azide
AP13278Pomalidomide 4-PEG3-Azide 474.5≥95% Pricing
AP12130Pomalidomide-PEG4-Azide518.53≥95% Pricing
AP13279Pomalidomide-PEG5-Azide590.6≥98% Pricing
AP13887Pomalidomide-PEG8-Azide694.7≥95% Pricing
Pomalidomide-PEG-Bromide
AP12997Pomalidomide-PEG3-Bromide512.36≥95% Pricing
Pomalidomide-PEG-NH-Boc
AP13828Pomalidomide-PEG3-NH-Boc548.6≥95% Pricing
Pomalidomide-PEG-Ph-NH2
AP13280Pomalidomide-PEG4-Ph-NH2540.6≥95% Pricing
THAL-SNS-032
AP14679THAL-SNS-032869.00≥95% Pricing
Thalidomide
AP13817Thalidomide258.2≥98% Pricing
AP139553-{5,7-dioxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}piperidine-2,6-dione259.22≥95% Pricing
AP139565-Amino-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione273.24≥95% Pricing
AP121224-Hydroxy-thalidomide274.23≥95% Pricing
AP121294-Fluoro-thalidomide276.22≥95% Pricing
AP139572-(2,6-dioxopiperidin-3-yl)-5-fluoroisoindoline-1,3-dione276.22≥95% Pricing
AP139652-(2,6-Dioxopiperidin-3-yl)-5-ethynylisoindoline-1,3-dione282.25≥95% Pricing
AP139582-(2,6-Dioxopiperidin-3-Yl)-5,6-Difluoroisoindoline-1,3-Dione294.21≥95% Pricing
AP139642-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindoline-5-carboxylic acid302.24≥95% Pricing
AP139632-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindole-4-carboxylic acid302.24≥95% Pricing
AP12123Thalidomide-Acid332.27≥95% Pricing
AP139615-Bromo-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione337.12≥95% Pricing
AP139603-(4-Bromo-7-fluoro-1-oxoisoindolin-2-yl)piperidine-2,6-dione341.13≥95% Pricing
AP139662-Chloro-N-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)acetamide349.72≥95% Pricing
AP139622-(2,6-Dioxopiperidin-3-yl)-4-iodoisoindoline-1,3-dione384.13≥95% Pricing
AP139592-(2,6-Dioxopiperidin-3-yl)-5-fluoro-6-(piperazin-1-yl)isoindoline-1,3-dione hydrochloride 396.8≥95% Pricing
Thalidomide-5-amine
AP13929Thalidomide-5-(C6-amine)393.87≥95% Pricing
AP13930Thalidomide-5-(PEG2-amine)432.4≥95% Pricing
AP13931Thalidomide-5-(PEG4-amine)520.5≥95% Pricing
Thalidomide-Acid
AP12123Thalidomide-Acid332.27≥95% Pricing
AP13477Thalidomide-5-(PEG2-acid)461.4≥95% Pricing
AP13478Thalidomide-5-(PEG4-acid)549.5≥95% Pricing
Thalidomide-O-amido-PEG-NHBoc
AP13027Thalidomide-O-amido-PEG2-NHBoc562.58≥95% Pricing
AP13029Thalidomide-O-amido-propoxy-PEG2-C3-NHBoc634.68≥95% Pricing
Thalidomide-O-PEG-Acid
AP14113Thalidomide-O-Hexyl-Acid402.40≥95% Pricing
AP13443Thalidomide-O-PEG2-Acid434.4≥98% Pricing
AP13444Thalidomide-O-PEG4-Acid522.5≥98% Pricing
AP13001Thalidomide-O-PEG5-Acid566.56≥95% Pricing
AP13445Thalidomide-O-PEG6-Acid610.6≥98% Pricing
Thalidomide-O-PEG-alcohol
AP13014Thalidomide-O-PEG3-alcohol406.39≥95% Pricing
Thalidomide-O-PEG-Amine
AP13119Thalidomide-O-amido-C4-amine402.4≥95% Pricing
AP13874Thalidomide-O-PEG2-Amine405.4≥95% Pricing
AP14112Thalidomide-O-C6-Amine HCl409.90≥95% Pricing
AP13004Thalidomide-O-PEG2-Amine HCl salt441.87≥95% Pricing
AP13015Thalidomide-O-PEG3-amine449.46≥95% Pricing
AP12124Thalidomide-O-PEG4-Amine493.51≥95% Pricing
AP13120Thalidomide-O-amido-C4-amine TFA Salt516.43≥95% Pricing
AP12384Thalidomide-O-PEG5-amine537.56≥ (95%) Pricing
AP13023Thalidomide-O-amido-C6-amine TFA salt544.48≥95% Pricing
AP13028Thalidomide-O-amido-C8-NHBoc558.63≥95% Pricing
AP13022Thalidomide-O-amido-C8-amine TFA salt572.54≥95% Pricing
AP13020Thalidomide-O-amido-PEG2-amine TFA salt576.48≥95% Pricing
AP12385Thalidomide-O-PEG6-amine581.62≥ (95%) Pricing
AP13024Thalidomide-O-amido-PEG3-amine TFA salt620.54≥95% Pricing
AP13026Thalidomide-O-amido-propoxy-PEG2-C3-amine TFA salt648.59≥95% Pricing
AP13025Thalidomide-O-amido-PEG4-amine TFA salt664.59≥95% Pricing
Thalidomide-O-PEG-Azide
AP11576Thalidomide-O-PEG4-Azide519.51≥95% Pricing
AP12125Thalidomide-O-amido-PEG4-azide576.56≥95% Pricing
Thalidomide-O-PEG-CH2-Ald
AP13013Thalidomide-O-PEG2-CH2-Ald404.38≥95% Pricing
Thalidomide-O-PEG-NHS ester
AP13384Thalidomide-O-PEG2-NHS ester531.5≥98% Pricing
AP12126Thalidomide-O-PEG4-NHS ester619.58≥95% Pricing
AP13385Thalidomide-O-PEG6-NHS ester707.7≥98% Pricing
Thalidomide-O-PEG-Propargyl
AP13003Thalidomide-O-PEG2-Propargyl400.39≥95% Pricing
AP13002Thalidomide-O-PEG3-Propargyl444.44≥95% Pricing
AP12334Thalidomide-O-PEG4-Propargyl488.49≥95% Pricing
AP12127Thalidomide-O-amido-PEG4-propargyl545.55≥95% Pricing
Thalidomide-O-PEG-t-butyl ester
AP12128Thalidomide-O-PEG4-t-butyl ester578.62≥95% Pricing
Thalidomide-O-PEG-Tosyl
AP13816Thalidomide-O-PEG5-Tosyl648.6≥98% Pricing
VH-298
AP14678VH-298523.70≥95% Pricing
VHL Ligand 1
AP12131VHL Ligand 1 HCl salt467.03≥95% Pricing

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