SGC-CBP30 is a potent CREBBP/EP300 inhibitor with IC50s of 21 nM and 38 nM, respectively, in cell-free assays. The selectivity for CBP is 40-fold and 250-fold higher than the first BRD for BRD4 (BRD4) and BRD4, respectively. SGC-CBP30 accelerates FRAP recovery in cells at a concentration of 1 μM.
AxisPharm offers 5000+ PEG Linkers with high purity. Different kinds of PEG Reagents may be available by custom synthesis.
![l-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)-lHpyrazolo [3,4-d]pyrimidin-l-yl]-l-piperidinyl]-2-propyn-l-one](https://e1752fbe.rocketcdn.me/wp-content/uploads/AP14272-CAS-936563-91-6-1-e1686054563587.png)