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HomePolyethylene Glycol PEG LinkersPROTAC LinkerBET Inhibitors GSK 5959
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GSK 5959

Catalog #: AP14260
Name: GSK 5959
Chemical Formula: C22H26N4O3
Molecular Weight: 394.50
CAS: 901245-65-6
Purity: ≥95%
Availability: In Stock

GSK 5959

$140.00 – $280.00

UnitPriceQuantity
10 mg$140
25 mg$280

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SKU: AP14260 Category: BET Inhibitors
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  • Description
  • Synonyms
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Description

GSK-5959 CAS:901245-65-6 is a potent, selective and cell-permeable BRPF1 bromodomain inhibitor with IC50 ~80 nM. More than 100-fold selectivity for BRPF1 (IC50 = 80 nM) over other 35 bromodomains including BRPF2/3 and BET family bromodomains. Inhibits the interaction of BRPF1 with histone H3.3, which is involved in epigenetic regulation of gene expression and has been implicated in human cancer.

AxisPharm offers 5000+ PEG Linkers with high purity. Different kinds of PEG Reagents may be available by custom synthesis.

Synonyms
  • 901245-65-6
  • GSK-5959
  • GSK 5959
  • GSK5959
  • N-[2,3-Dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxybenzamide
  • N-(1,3-dimethyl-2-oxo-6-piperidin-1-ylbenzimidazol-5-yl)-2-methoxybenzamide
  • N-[1,3-Dimethyl-2-Oxo-6-(Piperidin-1-Yl)-2,3-Dihydro-1h-Benzimidazol-5-Yl]-2-Methoxybenzamide
  • N-(1,3-dimethyl-2-oxo-6-(piperidin-1-yl)-2,3-dihydro-1H-benzo[d]imidazol-5-yl)-2-methoxybenzamide
  • N-(1,3-dimethyl-2-oxo-6-piperidin-1-yl-2,3-dihydro-1H-benzimidazol-5-yl)-2-methoxybenzamide
  • N-[1,3-dimethyl-2-oxo-6-(piperidin-1-yl)-2,3-dihydro-1H-1,3-benzodiazol-5-yl]-2-methoxybenzamide
Shipping & Delivery
Ships within: 24 hours
Storage condition: -20 ° C
Shipping: Ambient Temperature

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